K Nearest Neighbor and 3D QSAR Analysis of Thiazolidinone Derivatives as Antitubercular Agents

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Synthesis of Some 4-Thiazolidinone Derivatives as Antitubercular Agents

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synthesis of some 4-thiazolidinone derivatives as antitubercular agents

substituted schiff's bases 2a-o prepared by the treatment of 2-amino-4-(?-methoxyiminocarbomethoxymethyl)-thiazole 1 with different aromatic aldehydes, on cyclocondensation with mercaptoaceticacid and mercaptopropionicacid in dry benzene furnished desired thiazolidinones of type 3a-o and 4a-j, respectively. the structure of the compounds have been assigned on the basis of elemental analyse...

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3d qsar studies of 1,3,4-oxadiazole derivatives as antimycobacterial agents

recently several 1,3,4-oxadiazole derivatives were identified as potentially active antimycobacterial agents. various 5-aryl-2-thio-1,3,4-oxadiazoles have been reported having good antimycobacterial activity against mycobacterium tuberculosis h37rv (atcc 27294). in this paper we report 3d qsar studies for the 41 molecules of 1,3,4-oxadiazoles by using k-nearest neighbor molecular field analysis...

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ژورنال

عنوان ژورنال: Journal of Pharmaceutical Research

سال: 2016

ISSN: 2454-8405,0973-7200

DOI: 10.18579/jpcrkc/2016/15/3/103037